4-Cyanophenylboronic acid → 4-(6-Bromoimidazo[1,2-a]pyridin-3-yl)benzonitrile

Participants

Reaction Steps

The title compound, light brown solid (0.47 g, 73%), MS (ISP) m/z=298.4 [(M+H)+], mp 176° C., was prepared in accordance with the general method of intermediate E from commercially available 6-bromo-3-iodoimidazo[1,2-a]pyridine (0.7 g, 2.17 mmol) and commercially available 4-cyano-phenylboronic acid (0.36 g, 2.38 mmol).

Provenance & Evidence