4-(Methanesulfonyl)phenylboronic acid → 6-Bromo-3-(4-methanesulfonyl-phenyl)-imidazo[1,2-a]pyridine

Participants

Reaction Steps

The title compound, brown solid (0.53 g, 69%), MS (ISP) m/z=353.4 [(M+H)+], mp 194° C., was prepared in accordance with the general method of intermediate E from commercially available 6-bromo-3-iodoimidazo[1,2-a]pyridine (0.7 g, 2.17 mmol) and commercially available 4-methanesulfonyl-phenylboronic acid (0.48 g, 2.38 mmol).

Provenance & Evidence