5-Nitroindazole → 1H-Indazol-5-amine
Reaction equation
[N+:1]([C:4]1[CH:5]=[C:6]2[C:10](=[CH:11][CH:12]=1)[NH:9][N:8]=[CH:7]2)([O-])=O>[Pd]>[NH2:1][C:4]1[CH:5]=[C:6]2[C:10](=[CH:11][CH:12]=1)[NH:9][N:8]=[CH:7]2Participants
3
Reactant 1
Product 1
Reagents, catalysts & solvents 1
Procedure
By referring to the Step 6 of Example 1, 5-nitroindazole (5.0 g, 30.7 mmol), Pd/C (1.2 g), were used to obtain a product (2.6 g, 62.6%).
Sources & evidence
- ORD record
- ord-f599d3e385c7401d87a3d2decd23f378
- Source dataset
- uspto-grants-2016_04
- Patent number
- US09315513B2
Reaction notes
Loading…