HCID 86726370, compound → HCID 73438453, compound

HRID 629795Notes

Reaction equation

HRID 629795 reaction equation
[F:1][C:2]1[CH:7]=[CH:6][C:5]([C@@H:8]([C:13]2[CH:18]=[CH:17][N:16]=[CH:15][C:14]=2[F:19])[CH2:9][C:10]([OH:12])=O)=[CH:4][CH:3]=1.[NH2:20][C:21]1[CH:51]=[CH:50][CH:49]=[C:48]([F:52])[C:22]=1[CH2:23][CH2:24][C@H:25]1[O:30][CH2:29][C@@H:28]([CH2:31][O:32][C:33](=[O:40])[NH:34][CH2:35][C:36]([F:39])([F:38])[F:37])[N:27](C(OC(C)(C)C)=O)[CH2:26]1>>[F:39][C:36]([F:37])([F:38])[CH2:35][NH:34][C:33](=[O:40])[O:32][CH2:31][C@@H:28]1[CH2:29][O:30][C@H:25]([CH2:24][CH2:23][C:22]2[C:21]([NH:20][C:10](=[O:12])[CH2:9][C@@H:8]([C:5]3[CH:4]=[CH:3][C:2]([F:1])=[CH:7][CH:6]=3)[C:13]3[CH:18]=[CH:17][N:16]=[CH:15][C:14]=3[F:19])=[CH:51][CH:50]=[CH:49][C:48]=2[F:52])[CH2:26][NH:27]1

Participants

3

Reactant 2

HCID 86726370HCID 86726370, compoundHCID 86726409HCID 86726409, compound

Product 1

HCID 73438453HCID 73438453, compound

Procedure

The title compound was prepared from the product of step 1 and the product of step 4 of Example 99 using the procedures given in steps 8 and 9 of Example 89. MS (ES) m/z=625.5 (M+H)+.

Sources & evidence

ORD record
ord-68530e885b594b269549ddd5a618e3f8
Source dataset
uspto-grants-2016_04
Patent number
US09315475B2

Reaction notes

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