HuagongsheHuagongshe Chemistry Print Report · For research reference only
Phenylboronic Acid → (3-(Methylthio)-1-(5-phenylpyrimidin-2-yl)-1H-indol-6-yl)(morpholino)methanone
Participants
| Role | Name | HCID | Charge |
|---|---|---|---|
| Reactant | Phenylboronic Acid | HCID 66827 | — |
| Reactant | (1-(5-Bromopyrimidin-2-yl)-3-(methylthio)-1H-indol-6-yl)(morpholino)methanone | HCID 118666053 | — |
| Product | (3-(Methylthio)-1-(5-phenylpyrimidin-2-yl)-1H-indol-6-yl)(morpholino)methanone | HCID 118666064 | — |
Reaction Steps
Obtained according to general procedure 1 from (1-(5-bromopyrimidin-2-yl)-3-(methylthio)-1H-indol-6-yl)(morpholino)methanone (0.7 g, 1.616 mmol) and phenyl boronic acid (0.232 g, 1.939 mmol). Yield: 0.5 g (72% of theory)
Provenance & Evidence
| DOI | 10.6084/m9.figshare.5104873.v1 |
|---|---|
| Patent number | US09315490B2 |
| Source dataset | uspto-grants-2016_04 |
| ORD ID | ord-28495f93664c4c0aa5bce5db98c3f870 |
| Source note | uspto-grants-2016_04 |