3-(1-Bromoethyl)-4-phenyl-1H-isochromen-1-one → 3-(1-(2,6-diamino-9H-purin-9-yl)ethyl)-4-phenyl-1H-isochromen-1-one

Participants

Reaction Steps

The title compound was made in a similar way as that of the compound of example 1 from 3-(1-bromoethyl)-4-phenyl-1H-isochromen-1-one (intermediate C7, 50 mg, 0.15 mmol) and 9H-purine-2,6-diamine (34 mg, 0.23 mmol) to give the title compound (19 mg, 31%).

Provenance & Evidence