HRID639275
反应详情
EQUATION
反应方程式
REACTANTS
反应物
PRODUCTS
生成物
PROCEDURE
实验过程
The title compound was synthesized from 2,2,2-trichloro-1-{10-[(4-chlorophenoxy)acetyl]-10,11-dihydro-5H-pyrrolo[2,1-c][1,4]benzodiazepin-3-yl}ethanone of Example 67 (0.3 mmol) and 2-amino-1-phenylethanol (2.2 eq.) in the manner of Example 68, m.p. 157-158° C. MS [(−)ESI, m/z]: 514.3 [M−H]−