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HuagongsheHuagongshe Chemistry Print Report · For research reference only
HRID 643415Generated: October 30, 2026

methyl 1H-indole-4-carboxylate → Methyl 2-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)-1H-indole-4-carboxylate

https://huagongshe.com/reaction/643415

Reaction equation

Participants

RoleNameHCIDCharge
Reactantmethyl 1H-indole-4-carboxylateHCID 2733668—
Reactant7-Chloro-2-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-YL)-1H-indoleHCID 53217211—
ProductMethyl 2-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)-1H-indole-4-carboxylateHCID 53217126—

Reaction Steps

Prepared according to a procedure analogous to that described for 7-chloro-2-(4,4,5,5-tetramethyl-[1,3,2]dioxaborolan-2-yl)-1H-indole using 1H-indole-4-carboxylic acid, methyl ester.

Provenance & Evidence

DOI10.6084/m9.figshare.5104873.v1
Patent numberUS07700594B2
Source datasetuspto-grants-2010_04
ORD IDord-b6413cb631864d418e635988d206a15e
Source noteuspto-grants-2010_04