HuagongsheHuagongshe Chemistry Print Report · For research reference only
tert-butyl (3R)-3-aminopiperidine-1-carboxylate → (R)-N-(Piperidin-3-yl)-1H-indazol-5-amine
Participants
| Role | Name | HCID | Charge |
|---|---|---|---|
| Reactant | tert-butyl (3R)-3-aminopiperidine-1-carboxylate | HCID 1501974 | — |
| Reactant | 5-Bromo-1-(4-methoxybenzyl)-1H-indazole | HCID 44240527 | — |
| Product | (R)-N-(Piperidin-3-yl)-1H-indazol-5-amine | HCID 44240125 | — |
Reaction Steps
Reaction of 5-bromo-1-(4-methoxybenzyl)-1H-indazole and (R)-tert-butyl 3-aminopiperidine-1-carboxylate using the method of Example 13 followed by deprotection using the method of Example 14 afforded the title compound.
Provenance & Evidence
| DOI | 10.6084/m9.figshare.5104873.v1 |
|---|---|
| Patent number | US08071779B2 |
| Source dataset | uspto-grants-2011_12 |
| ORD ID | ord-63b5079ccf874144bf6180cc977bdaed |
| Source note | uspto-grants-2011_12 |