反应详情

Using general procedure 2 with [(R)-2-(2-fluoro-phenyl)-1-(methoxy-methyl-carbamoyl)-ethyl]-carbamic acid tert-butyl ester (3.5 g, 11 mmol) and N-tert-Butyl-4-chloro-2-methyl-benzamide (7.3 g, 32 mmol) followed by purification using silica gel flash column chromatography gives the title compound.

1. customfollowed by purification