反应详情

Using general procedure 2 with [(R)-2-(2-fluoro-phenyl)-1-(methoxy-methyl-carbamoyl)-ethyl]-carbamic acid tert-butyl ester (2.15 g, 6.6 mmol) and N-tert-butyl-2,5-dimethyl-benzamide (4.0 g, 20 mmol), followed by purification by silica gel flash column chromatography gives the title compound.

1. customfollowed by purification by silica gel flash column chromatography