N-(1-Cyano-piperidin-4-yl)-N-cyclopropyl-4-oxazol-5-yl-benzamide → N-Cyclopropyl-N-{1-[3-(4-fluoro-phenyl)-[1,2,4]oxadiazol-5-yl]-piperidin-4-yl}-4-oxazol-5-yl-benzamide

Participants

Reaction Steps

The title compound is prepared from N-(1-cyano-piperidin-4-yl)-N-cyclopropyl-4-oxazol-5-yl-benzamide and 4-fluoro-N-hydroxy-benzamidine following a procedure analogous to that described in Example 1. LC (method 6): tR=1.87 min; Mass spectrum (ESI+): m/z=474 [M+H]+.

Provenance & Evidence