N-(1-Cyano-piperidin-4-yl)-N-cyclopropyl-4-oxazol-5-yl-benzamide → N-Cyclopropyl-4-oxazol-5-yl-N-[1-(3-thiophen-3-yl-[1,2,4]oxadiazol-5-yl)-piperidin-4-yl]-benzamide

Participants

Reaction Steps

The title compound is prepared from N-(1-cyano-piperidin-4-yl)-N-cyclopropyl-4-oxazol-5-yl-benzamide and N-hydroxy-thiophene-3-carboxamidine following a procedure analogous to that described in Example 1. LC (method 6): tR=1.78 min; Mass spectrum (ESI+): m/z=462 [M+H]+.

Provenance & Evidence