N-(1-Cyano-piperidin-4-yl)-N-cyclopropyl-4-oxazol-5-yl-benzamide → 5-{4-[Cyclopropyl-(4-oxazol-5-yl-benzoyl)-amino]-piperidin-1-yl}-[1,2,4]oxadiazole-3-carboxylic acid ethyl ester

Participants

Reaction Steps

The title compound is prepared from N-(1-cyano-piperidin-4-yl)-N-cyclopropyl-4-oxazol-5-yl-benzamide and hydroxyamino-imino-acetic acid ethyl ester following a procedure analogous to that described in Example 1. LC (method 3): tR=1.77 min; Mass spectrum (ESI+): m/z=452 [M+H]+.

Provenance & Evidence