反应详情

In analogy to the procedure described for the preparation of example 1, (rac)-N-(4-bromo-6,7-dihydro-5H-cyclopenta[c]pyridin-7-yl)propionamide (intermediate A-4) was reacted with 4-chloro-3-fluorophenylboronic acid to give the title compound as grey solid in 87% yield. MS: 319.1 (M+H+, 1Cl).