反应详情

In analogy to the procedure described for the preparation of (rac)-cyclopropanesulfonic acid [4-(4-trifluoromethyl-phenyl)-6,7-dihydro-5H-[2]pyrindin-7-yl]-amide (example 94), replacing cyclopropanesulfonyl chloride with propane-1-sulfonyl chloride. The title compound was obtained as a light brown oil in 5% yield. MS: 385.5 (M+H)+.