HuagongsheHuagongshe Chemistry Print Report · For research reference only
methyl (R)-7-amino-2,3,3a,4-tetrahydro-1H-benzo[b]pyrrolo[1,2-d][1,4]oxazine-6-carboxylate → Methyl (S)-7-amino-2,3,3a,4-tetrahydro-1H-benzo[b]pyrrolo[1,2-d][1,4]oxazine-6-carboxylate
Participants
| Role | Name | HCID | Charge |
|---|---|---|---|
| Reactant | methyl (R)-7-amino-2,3,3a,4-tetrahydro-1H-benzo[b]pyrrolo[1,2-d][1,4]oxazine-6-carboxylate | HCID 86712109 | — |
| Reactant | methyl 6-amino-3-bromo-2-((S)-1-pyrrolidin-2-ylmethoxy)benzoate | HCID 86712113 | — |
| Product | Methyl (S)-7-amino-2,3,3a,4-tetrahydro-1H-benzo[b]pyrrolo[1,2-d][1,4]oxazine-6-carboxylate | HCID 86712112 | — |
Reaction Steps
Prepared by proceeding in a similar manner to Intermediate 6, starting from methyl 6-amino-3-bromo-2-((S)-1-pyrrolidin-2-ylmethoxy)benzoate (Intermediate 14).
Provenance & Evidence
| DOI | 10.6084/m9.figshare.5104873.v1 |
|---|---|
| Patent number | US09187494B2 |
| Source dataset | uspto-grants-2015_11 |
| ORD ID | ord-de4fb148b73a4262a98cb60fbfc66ea7 |
| Source note | uspto-grants-2015_11 |