HuagongsheHuagongshe Chemistry Print Report · For research reference only
HCID 57360953, compound → Ethyl 6-((5-chloro-2-(3-(3-fluorophenoxy)azetidin-1-yl)nicotinamido)methyl)nicotinate
Participants
| Role | Name | HCID | Charge |
|---|---|---|---|
| Reactant | HCID 57360953 | HCID 57360953 | — |
| Reactant | 5-Chloro-2-(3-(3-fluorophenoxy)azetidin-1-yl)nicotinic acid | HCID 67958861 | — |
| Product | Ethyl 6-((5-chloro-2-(3-(3-fluorophenoxy)azetidin-1-yl)nicotinamido)methyl)nicotinate | HCID 67958672 | — |
Reaction Steps
The title compound (D158) (59 mg) was prepared according to the experimental procedure described in Description 144 starting from 5-chloro-2-(3-(3-fluorophenoxy)azetidin-1-yl)nicotinic acid (D103) (50 mg, 0.154 mmol) and ethyl 6-(aminomethyl)nicotinate hydrochloride (33.56 mg, 0.154 mmol, commercially available at Chemimpex#23882).
Provenance & Evidence
| DOI | 10.6084/m9.figshare.5104873.v1 |
|---|---|
| Patent number | US08828987B2 |
| Source dataset | uspto-grants-2014_09 |
| ORD ID | ord-c63c9e4bb7c142c0996d960c00ff6578 |
| Source note | uspto-grants-2014_09 |