(1-ethyl-1H-indazol-5-yl)methanamine → HCID 66837826, compound
Reaction equation
[Cl:1][C:2]1[CH:3]=[C:4]([CH:10]=[CH:11][C:12]=1[S:13](Cl)(=[O:15])=[O:14])[C:5]([O:7][CH2:8][CH3:9])=[O:6].[CH2:17]([N:19]1[C:27]2[C:22](=[CH:23][C:24]([CH2:28][NH2:29])=[CH:25][CH:26]=2)[CH:21]=[N:20]1)[CH3:18]>>[Cl:1][C:2]1[CH:3]=[C:4]([CH:10]=[CH:11][C:12]=1[S:13](=[O:15])(=[O:14])[NH:29][CH2:28][C:24]1[CH:23]=[C:22]2[C:27](=[CH:26][CH:25]=1)[N:19]([CH2:17][CH3:18])[N:20]=[CH:21]2)[C:5]([O:7][CH2:8][CH3:9])=[O:6]Participants
3
Procedure
The titled compound was prepared according to the procedure described in step-1 of Example 1 from ethyl 3-chloro-4-(chlorosulfonyl)benzoate and (1-ethyl-1H-indazol-5-yl)methanamine (step-3 of Example 14).
Sources & evidence
- ORD record
- ord-e4cdd6ba81934f72ab04c892c6ceb34d
- Source dataset
- uspto-grants-2014_09
- Patent number
- US08829026B2
Reaction notes
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