N-(3-Aminopropyl)morpholine → HCID 24738672, compound

Participants

Reaction Steps

As described for Example 11b, 2-(5-methyl-3-phenyl-isoxazol-4-yl)-imidazo[1,2-a]pyridine-7-carboxylic acid (96 mg, 0.3 mmol) was converted, using N-(3-aminopropyl)morpholine instead of aminomethylcyclopropane, to the title compound (102 mg, 76%) which was obtained as an off-white foam. MS: m/e=446.3 [M+H]+.

Provenance & Evidence