戻る
化工社化工社 化学情報印刷レポート · 研究参考用
HRID 736166作成日：2026年10月25日

Benzoic acid, 2-chloro-5-[(methylamino)sulfonyl]- → 3-[4-(4-Acetyl-2-fluoro-phenyl)-piperazine-1-carbonyl]-4-chloro-N-methyl-benzenesulfonamide

https://huagongshe.com/reaction/736166

反応式

関与物質

役割名称HCID仕込み量
反応物Benzoic acid, 2-chloro-5-[(methylamino)sulfonyl]-HCID 111724—
反応物1-(3-Fluoro-4-piperazin-1-ylphenyl)ethanoneHCID 685610—
生成物3-[4-(4-Acetyl-2-fluoro-phenyl)-piperazine-1-carbonyl]-4-chloro-N-methyl-benzenesulfonamideHCID 59793606—

反応手順

The title compound was prepared according to the procedure described for example K/step 2 from 1-(3-Fluoro-4-piperazin-1-yl-phenyl)-ethanone and 2-Chloro-5-methylsulfamoyl-benzoic acid (CAS: 68901-09-7; BE 620741) (69%, light yellow foam, MS (m/e): 452.1 (M−H, 100%)

情報源と証拠

DOI10.6084/m9.figshare.5104873.v1
特許番号US07595314B2
出典データセットuspto-grants-2009_09
ORD IDord-2f8988f3123848b0a27f20c03009b638
出典メモuspto-grants-2009_09