Hydroxylamine → HCID 86607878, compound

Participants

Reaction Steps

According to the procedure of Example 17, Step 5, the reaction of 122 mg of cis-1-(tert-butoxycarbonyl)-4-[({4-[(2-methylquinolin-4-yl)methoxy]phenyl}sulfonyl)amino]pyrrolidine-3-carboxylic acid with hydroxylamine provided 104 mg (81% yield) of tert-butyl cis-3-[(hydroxyamino)carbonyl]-4-[({4-[(2-methylquinolin-4-yl)methoxy]phenyl}sulfonyl)amino]pyrrolidine-1-carboxylate. MS: 557.3 (M+H)+

Provenance & Evidence