3-(Aminomethyl)benzeneboronic acid, N-BOC protected → [3-(2-Amino-6-methyl-[1,2,4]triazolo[1,5-a]pyridin-8-yl)-benzyl]-carbamic acid tert-butyl ester
Reaction equation
[Br:1][c:2]1[c:3]2[n:4]([cH:5][c:6]([CH3:8])[cH:7]1)[n:9][c:10]([NH2:12])[n:11]2.[C:13]([CH3:14])([CH3:15])([CH3:16])[O:17][C:18](=[O:19])[NH:20][CH2:21][c:22]1[cH:23][c:24]([B:28]([OH:29])[OH:30])[cH:25][cH:26][cH:27]1>>[c:2]1(-[c:24]2[cH:23][c:22]([CH2:21][NH:20][C:18]([O:17][C:13]([CH3:14])([CH3:15])[CH3:16])=[O:19])[cH:27][cH:26][cH:25]2)[c:3]2[n:4]([cH:5][c:6]([CH3:8])[cH:7]1)[n:9][c:10]([NH2:12])[n:11]2Participants
3
Sources & evidence
- ORD record
- ord-2ad62cff5eaa40c1b09ffbc575eadff7
- Source dataset
- Test data from https://doi.org/10.1039/C8SC04228D
Reaction notes
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