5-(4-Methylbenzyl)-benzofuran-2-ylboronic acid → Methyl 1-(3-fluoro-4-(5-(4-methylbenzyl)benzofuran-2-yl)benzyl)azetidine-3-carboxylate
Reaction equation
[Br:21][c:22]1[c:23]([F:37])[cH:24][c:25]([CH2:26][N:27]2[CH2:28][CH:29]([C:31](=[O:32])[O:33][CH3:34])[CH2:30]2)[cH:35][cH:36]1.[CH3:1][c:2]1[cH:3][cH:4][c:5]([CH2:6][c:7]2[cH:8][cH:9][c:10]3[c:11]([cH:12][c:13]([B:15]([OH:16])[OH:17])[o:14]3)[cH:18]2)[cH:19][cH:20]1>>[CH3:1][c:2]1[cH:3][cH:4][c:5]([CH2:6][c:7]2[cH:8][cH:9][c:10]3[c:11]([cH:12][c:13](-[c:22]4[c:23]([F:37])[cH:24][c:25]([CH2:26][N:27]5[CH2:28][CH:29]([C:31](=[O:32])[O:33][CH3:34])[CH2:30]5)[cH:35][cH:36]4)[o:14]3)[cH:18]2)[cH:19][cH:20]1Participants
3
Sources & evidence
- ORD record
- ord-15f99d2f02d34fa8bc563976995732b3
- Source dataset
- Test data from https://doi.org/10.1039/C8SC04228D
Reaction notes
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