Cyclopentylamine → HCID 77750349, compound

HRID 840706Notes

Reaction equation

[OH:1][CH:2]1[CH:6]([OH:7])[CH:5]([N:8]2[C:12]3[N:13]=[C:14]([S:27][CH3:28])[N:15]=[C:16]([NH:17][CH:18]4[CH2:20][CH:19]4[C:21]4[CH:26]=[CH:25][CH:24]=[CH:23][CH:22]=4)[C:11]=3[N:10]=[N:9]2)[CH2:4][CH:3]1[C:29]([NH:31][C:32]1[CH:37]=[CH:36][CH:35]=[CH:34]C=1)=[O:30].C1(N)CCCC1>>[CH:32]1([NH:31][C:29]([CH:3]2[CH2:4][CH:5]([N:8]3[C:12]4[N:13]=[C:14]([S:27][CH3:28])[N:15]=[C:16]([NH:17][CH:18]5[CH2:20][CH:19]5[C:21]5[CH:22]=[CH:23][CH:24]=[CH:25][CH:26]=5)[C:11]=4[N:10]=[N:9]3)[CH:6]([OH:7])[CH:2]2[OH:1])=[O:30])[CH2:37][CH2:36][CH2:35][CH2:34]1

Participants

Reactant 2

HCID 2906Cyclopentylamine

HCID 77750267HCID 77750267, compound

Product 1

HCID 77750349HCID 77750349, compound

Procedure

The title compound was prepared according to the method of example 1, step d) using the product of Example 20, step b) and cyclopentylamine, followed by deprotection according to the method of example 1, step e).

Sources & evidence

ORD record: ord-684df9ace07d4c808a4b163c81c8f68c
Source dataset: uspto-grants-2002_04
DOI: 10.6084/m9.figshare.5104873.v1
Patent number: US06369064B1

Reaction notes

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