(3-Bromophenyl)boronic acid → 7-(3-bromophenoxy)-2,3-dihydro-1H-pyrrolo[2,1-c][1,2,4]benzothiadiazine 5,5-dioxide

HRID 851886Notes

Reaction equation

HRID 851886 reaction equation
[Br:1][C:2]1[CH:3]=[C:4](B(O)O)[CH:5]=[CH:6][CH:7]=1.[O:11]=[S:12]1(=[O:33])[C:17]2[CH:18]=[C:19]([O:22]C3C=C(O)C=CC=3)[CH:20]=[CH:21][C:16]=2[N:15]2[CH2:30][CH2:31][CH2:32][C:14]2=[N:13]1>>[Br:1][C:2]1[CH:3]=[C:4]([CH:5]=[CH:6][CH:7]=1)[O:22][C:19]1[CH:20]=[CH:21][C:16]2[N:15]3[CH2:30][CH2:31][CH2:32][C:14]3=[N:13][S:12](=[O:33])(=[O:11])[C:17]=2[CH:18]=1

Participants

3

Reactant 2

HCID 2734318(3-Bromophenyl)boronic acidHCID 12157386HCID 12157386, compound

Product 1

HCID 694145897-(3-bromophenoxy)-2,3-dihydro-1H-pyrrolo[2,1-c][1,2,4]benzothiadiazine 5,5-dioxide

Procedure

The procedure is as in Step B of Example 1, using as starting materials (3-bromophenyl)boronic acid and the product obtained in Step A of Example 1.

Sources & evidence

ORD record
ord-07119cfa10f0491d89a01c52a138fae8
Source dataset
uspto-grants-2007_08
Patent number
US07253163B2

Reaction notes

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