4-Hydroxybenzoic Acid → HCID 10223901, compound

HRID 854309Notes

Reaction equation

HRID 854309 reaction equation
[F:1][C:2]1[CH:7]=[CH:6][C:5]([CH2:8][CH2:9][S:10]([N:13]2[CH2:18][CH2:17][CH:16]([CH2:19][NH2:20])[CH2:15][CH2:14]2)(=[O:12])=[O:11])=[CH:4][CH:3]=1.[OH:21][C:22]1[CH:30]=[CH:29][C:25]([C:26](O)=[O:27])=[CH:24][CH:23]=1>>[F:1][C:2]1[CH:7]=[CH:6][C:5]([CH2:8][CH2:9][S:10]([N:13]2[CH2:14][CH2:15][CH:16]([CH2:19][NH:20][C:26](=[O:27])[C:25]3[CH:29]=[CH:30][C:22]([OH:21])=[CH:23][CH:24]=3)[CH2:17][CH2:18]2)(=[O:11])=[O:12])=[CH:4][CH:3]=1

Participants

3

Reactant 2

HCID 1354-Hydroxybenzoic AcidHCID 22135614HCID 22135614, compound

Product 1

HCID 10223901HCID 10223901, compound

Procedure

N-{1-[2-(4-Fluoro-phenyl)-ethanesulfonyl]-piperidin-4-ylmethyl}-4-hydroxy-benzamide was prepared from C-{1-[2-(4-fluoro-phenyl)-ethanesulfonyl]-piperidin-4-yl}-methylamine and 4-hydroxybenzoic acid as described above in EXAMPLE 1, Step 2

Sources & evidence

ORD record
ord-179f7ddbc2474f849d151a7ef79cc75f
Source dataset
uspto-grants-2007_08
Patent number
US07259157B2

Reaction notes

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