Thiophene-3-boronic acid → HCID 10249400, compound

Participants

Reaction Steps

Cross-coupling of 2-(6-chloropyridin-3-yl)-3-cyclopentyl-N-thiazol-2-ylpropionamide (EXAMPLE 1, 100 mg, 297 μmol) with thiophene-3-boronic acid (100 mg, 781 μmol), utilising a procedure similar to that described above for EXAMPLE 2, furnished the title compound: RTA=3.83 min; m/z (ES+)=384.2 [M+H]+.

Provenance & Evidence