2-Morpholinoethanol → HCID 66850566, compound

HRID 873688Notes

Reaction equation

HRID 873688 reaction equation
[OH:1][CH2:2][CH2:3][N:4]1[CH2:9][CH2:8][O:7][CH2:6][CH2:5]1.CN(C)CCO[C:15]1[CH:20]=[C:19]([B:21]([OH:23])[OH:22])[CH:18]=[CH:17][N:16]=1>>[N:4]1([CH2:3][CH2:2][O:1][C:15]2[CH:20]=[C:19]([B:21]([OH:23])[OH:22])[CH:18]=[CH:17][N:16]=2)[CH2:9][CH2:8][O:7][CH2:6][CH2:5]1

Participants

3

Reactant 2

HCID 611632-MorpholinoethanolHCID 66850324HCID 66850324, compound

Product 1

HCID 66850566HCID 66850566, compound

Procedure

[2-(2-Morpholin-4-yl-ethoxy)-4-pyridinyl]-boronic acid is prepared from N-(2-hydroxyethyl)-morpholine according to the procedure described for the preparation of [2-(2-dimethylamino-ethoxy)-4-pyridinyl]-boronic acid. MS (m/z): 253 (M+1).

Sources & evidence

ORD record
ord-6049bfa8edd14097845c9f5edd0eac1f
Source dataset
uspto-grants-2015_03
Patent number
US08975439B2

Reaction notes

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