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HuagongsheHuagongshe Chemistry Print Report · For research reference only
HRID 881317Generated: November 1, 2026

5-(4,4,5,5-Tetramethyl-1,3,2-dioxaborolan-2-yl)pyridin-2-amine → HCID 58234093, compound

https://huagongshe.com/reaction/881317

Reaction equation

Participants

RoleNameHCIDCharge
Reactant5-(4,4,5,5-Tetramethyl-1,3,2-dioxaborolan-2-yl)pyridin-2-amineHCID 2756555—
ReactantHCID 86623520HCID 86623520—
ProductHCID 58234093HCID 58234093—

Reaction Steps

1-(4-((2-Chloro-4-morpholinothieno[2,3-d]pyrimidin-6-yl)methyl)piperazin-1-yl)-2-hydroxyethanone (265 mg) was reacted with 5-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)pyridin-2-amine via General Procedure A to give 16.5 mg of 181. MS (Q1) 470.2 (M)+

Provenance & Evidence

DOI10.6084/m9.figshare.5104873.v1
Patent numberUS08993563B2
Source datasetuspto-grants-2015_03
ORD IDord-3ed2c47877044ef08ee713f8ac3ab05f
Source noteuspto-grants-2015_03