4-((5-Fluoropyridin-2-yl)methoxy)pyridin-2(1H)-one → tert-Butyl 7,9-dimethyl-2-(4-((5-fluoropyridin-2-yl)methoxy)-2-oxopyridin-1(2H)-yl)-5,7,8,9-tetrahydro-6H-pyrido[3',4':4,5]pyrrolo[2,3-b]pyridine-6-carboxylate

Beteiligte Stoffe

Reaktionsschritte

tert-Butyl 2-bromo-7,9-dimethyl-5,7,8,9-tetrahydro-6H-pyrido[3′,4′:4,5]pyrrolo[2,3-b]pyridine-6-carboxylate (200 mg, 0.520 mmol) and 4-((5-fluoropyridin-2-yl)methoxy)pyridin-2(1H)-one (115 mg, 0.520 mmol) were reacted following the procedure for Example 2 (step e) to provide the title compound (198 mg, 73%) as a yellow oil: ESI MS m/z 520 [M+H]+.

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