p-Chlorophenylboric acid → HCID 59691690, compound

HRID 898609Notes

Reaction equation

HRID 898609 reaction equation
Br[C:2]1[CH:7]=[CH:6][C:5]([NH:8][CH2:9][C:10]([NH:12][C:13]2[CH:18]=[CH:17][C:16]([CH2:19][N:20]([CH3:22])[CH3:21])=[CH:15][CH:14]=2)=[O:11])=[CH:4][CH:3]=1.[Cl:23][C:24]1[CH:29]=[CH:28][C:27](OB(O)O)=[CH:26][CH:25]=1>>[Cl:23][C:24]1[CH:29]=[CH:28][C:27]([C:2]2[CH:7]=[CH:6][C:5]([NH:8][CH2:9][C:10]([NH:12][C:13]3[CH:18]=[CH:17][C:16]([CH2:19][N:20]([CH3:22])[CH3:21])=[CH:15][CH:14]=3)=[O:11])=[CH:4][CH:3]=2)=[CH:26][CH:25]=1

Participants

3

Reactant 2

HCID 17810664p-Chlorophenylboric acidHCID 688767692-[(4-Bromophenyl)amino]-N-[4-[(dimethylamino)methyl]phenyl]acetamide

Product 1

HCID 59691690HCID 59691690, compound

Procedure

Prepared analogously to Example 130a starting from 2-(4-bromo-phenylamino)-N-(4-dimethylaminomethyl-phenyl)-acetamide (Example 163a) and 4-chloro-phenyl-boric acid.

Workup

  1. customPrepared analogously to Example 130a

Sources & evidence

ORD record
ord-abe6a09df0fd4a52bedfb38e813c5d57
Source dataset
uspto-grants-2008_04
Patent number
US07351719B2

Reaction notes

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