N-bromobutanimide → HCID 67388007, compound

Participants

Reaction Conditions

Reaction Steps

A mixture of 3-(7-methoxy-1,3-benzoxazol-2-yl)pyridin-2-amine (85 mg) and 1-bromopyrrolidine-2,5-dione (69.0 mg) in THF (2 ml) was stirred at 25° C. for 1 hour. The reaction mixture was concentrated to dryness and the resulting solid was triturated with water to give a solid which was collected by filtration and dried under vacuum to give 5-bromo-3-(7-methoxy-1,3-benzoxazol-2-yl)pyridin-2-amine (120 mg) as a solid.

Provenance & Evidence