HCID 10396998, compound → HCID 69121086, compound

HRID 915261Notes

Reaction equation

HRID 915261 reaction equation
[CH:1]1([C:6]([OH:18])([C:10]2[CH:15]=[CH:14][C:13]([O:16][CH3:17])=[CH:12][CH:11]=2)[C:7]([OH:9])=[O:8])[CH2:5][CH2:4][CH2:3][CH2:2]1.[CH:19]12[CH2:24][CH:23]1[CH2:22][N:21]([CH2:25][C:26]#[C:27][CH2:28]O)[CH2:20]2>>[C@@H:19]12[CH2:24][C@@H:23]1[CH2:22][N:21]([CH2:25][C:26]#[C:27][CH2:28][O:8][C:7](=[O:9])[C:6]([C:10]1[CH:15]=[CH:14][C:13]([O:16][CH3:17])=[CH:12][CH:11]=1)([CH:1]1[CH2:5][CH2:4][CH2:3][CH2:2]1)[OH:18])[CH2:20]2

Participants

3

Procedure

The title compound was prepared by following the procedure described in Step-b of Example-3, using 2-cyclopentyl-2-hydroxy-2-(4-methoxyphenyl)acetic acid instead of 2-cyclopentyl-2-hydroxy-2-phenyl acetic acid and 4-(3-azabicyclo[3.1.0]hex-3-yl)-2-butynol instead of 4-(1,5-dimethyl-3-azabicyclo[3.1.0]hex-3-yl)-2-butynol.

Sources & evidence

ORD record
ord-b7c5edb5fe1244fc82ef30ebaf4d8e62
Source dataset
uspto-grants-2007_09
Patent number
US07265147B2

Reaction notes

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