O-Toluidine → HCID 118113874, compound

HRID 918850Notes

Reaction equation

HRID 918850 reaction equation
[NH2:1][C:2]1[C:3]([CH3:8])=[CH:4][CH:5]=[CH:6][CH:7]=1.[Br:9][C:10]1[CH:11]=[CH:12][C:13]2[N:14]([CH:16]=[C:17]([C:19](OCC)=[O:20])[N:18]=2)[CH:15]=1>>[Br:9][C:10]1[CH:11]=[CH:12][C:13]2[N:14]([CH:16]=[C:17]([C:19]([NH:1][C:2]3[CH:7]=[CH:6][CH:5]=[CH:4][C:3]=3[CH3:8])=[O:20])[N:18]=2)[CH:15]=1

Participants

3

Reactant 2

HCID 7242O-ToluidineHCID 7141939Ethyl 6-bromoimidazo[1,2-a]pyridine-2-carboxylate

Product 1

HCID 118113874HCID 118113874, compound

Procedure

The title compound was prepared by using procedures analogous to those described for the synthesis of Intermediate I, using o-toluidine and ethyl 6-bromoimidazo[1,2-a]pyridine-2-carboxylate as starting materials.

Sources & evidence

ORD record
ord-d5d218b93497463fb6a39aa1972420f0
Source dataset
uspto-grants-2016_03
Patent number
US09271969B2

Reaction notes

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