2,4-Dichloro-6-methylbenzylamine → HCID 118114001, compound

HRID 918861Notes

Reaction equation

HRID 918861 reaction equation
[Cl:1][C:2]1[CH:7]=[C:6]([Cl:8])[CH:5]=[C:4]([CH3:9])[C:3]=1[CH2:10][NH2:11].[Br:12][C:13]1[CH:14]=[CH:15][C:16]2[N:17]([CH:19]=[C:20]([C:22](OCC)=[O:23])[N:21]=2)[CH:18]=1>>[Br:12][C:13]1[CH:14]=[CH:15][C:16]2[N:17]([CH:19]=[C:20]([C:22]([NH:11][CH2:10][C:3]3[C:4]([CH3:9])=[CH:5][C:6]([Cl:8])=[CH:7][C:2]=3[Cl:1])=[O:23])[N:21]=2)[CH:18]=1

Participants

3

Procedure

The title compound was prepared by using procedures analogous to those described for the synthesis of Intermediate I, using (2,4-dichloro-6-methylphenyl)methanamine and ethyl 6-bromoimidazo[1,2-a]pyridine-2-carboxylate as starting materials.

Sources & evidence

ORD record
ord-0b8f904aceb34ac4878b8ad66fc05fe9
Source dataset
uspto-grants-2016_03
Patent number
US09271969B2

Reaction notes

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