HCID 23005388, compound → HCID 71061029, compound
Reaction equation
[NH2:1][C:2]1[N:16]=[CH:15][C:14](Br)=[CH:13][C:3]=1[C:4]([NH:6][C:7]1[CH:12]=[CH:11][N:10]=[CH:9][CH:8]=1)=[O:5].[C:18]1([CH3:33])[CH:23]=[CH:22][C:21]([C:24]2[CH:25]=[C:26](B(O)O)[CH:27]=[CH:28][CH:29]=2)=[CH:20][CH:19]=1>>[NH2:1][C:2]1[N:16]=[CH:15][C:14]([C:26]2[CH:25]=[C:24]([C:21]3[CH:20]=[CH:19][C:18]([CH3:33])=[CH:23][CH:22]=3)[CH:29]=[CH:28][CH:27]=2)=[CH:13][C:3]=1[C:4]([NH:6][C:7]1[CH:12]=[CH:11][N:10]=[CH:9][CH:8]=1)=[O:5]Participants
3
Procedure
Reaction of 2-amino-5-bromo-N-pyridin-4-yl-nicotinamide with [3-(p-tolyl)phenyl]-boronic acid gives the compound “A23”;
Workup
- customgives the compound “A23”
Sources & evidence
- ORD record
- ord-2f2f8c207d434317adc015e8d9e803e1
- Source dataset
- uspto-grants-2016_03
- Patent number
- US09273029B2
Reaction notes
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