hydrogen chloride CPME → 4-(benzoylamino)-N-(4-{trans-2-[(cyclopropylmethyl)amino]-cyclopropyl}phenyl)benzamide hydrochloride

Participants

Reaction Steps

tert-Butyl [trans-2-(4-{[4-(benzoylamino)benzoyl]amino}phenyl)cyclopropyl]-(cyclopropylmethyl)carbamate (98.0 mg) was dissolved in 4N hydrochloric acid/cyclopentyl methyl ether solution (1 mL), and the mixture was stirred at room temperature for 2 hr. The solvent was evaporated under reduced pressure. The residue was recrystallized from methanol/diisopropyl ether to give the title compound (44.6 mg).

Provenance & Evidence