HCID 90036013, compound → HCID 118341128, compound

Participants

Reaction Steps

The title compound, off-white solid (68 mg, 80%), MS (ISP) m/z=342.5 [(M+H)+], mp 196° C., was prepared in accordance with the general method of example 1 from 6-bromo-8-chloro-10-methyl-3,4-dihydro-2H-pyrazino[1,2-a]indol-1-one (intermediate 12) (78.4 mg, 0.25 mmol) and commercially available 6-methoxy-pyridin-3-ylphenylboronic acid (49.7 mg, 0.325 mmol).

Provenance & Evidence