6-(3-Chlorophenyl)picolinic acid → HCID 71105541, compound

HRID 927369Notes

Reaction equation

HRID 927369 reaction equation
[Cl:1][C:2]1[CH:3]=[C:4]([C:8]2[N:13]=[C:12]([C:14]([OH:16])=O)[CH:11]=[CH:10][CH:9]=2)[CH:5]=[CH:6][CH:7]=1.[CH3:17][C:18]([NH2:25])([C:20]1[O:21][CH:22]=[N:23][N:24]=1)[CH3:19]>>[CH3:17][C:18]([NH:25][C:14]([C:12]1[CH:11]=[CH:10][CH:9]=[C:8]([C:4]2[CH:5]=[CH:6][CH:7]=[C:2]([Cl:1])[CH:3]=2)[N:13]=1)=[O:16])([C:20]1[O:21][CH:22]=[N:23][N:24]=1)[CH3:19]

Participants

3

Reactant 2

HCID 247301356-(3-Chlorophenyl)picolinic acidHCID 84647948HCID 84647948, compound

Product 1

HCID 71105541HCID 71105541, compound

Procedure

The title compound was synthesized in analogy to Example 1, using 6-(3-chlorophenyl)-2-pyridinecarboxylic acid (CAN 863704-38-5) and 1-methyl-1-[1,3,4]oxadiazol-2-yl-ethylamine as starting materials, MS (LC/MS): 343.0 [M+H]+.

Sources & evidence

ORD record
ord-fe17a6690b674dad9ff5cd53d9811dc4
Source dataset
uspto-grants-2016_03
Patent number
US09290451B2

Reaction notes

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