HuagongsheHuagongshe Chemistry Print Report · For research reference only
2-(5-Methyl-1,2,4-oxadiazol-3-yl)propan-2-amine → 5-Cyclopentyl-6-cyclopropylmethoxy-pyridine-2-carboxylic acid [1-methyl-1-(5-methyl-[1,2,4]oxadiazol-3-yl)-ethyl]-amide
Participants
| Role | Name | HCID | Charge |
|---|---|---|---|
| Reactant | 2-(5-Methyl-1,2,4-oxadiazol-3-yl)propan-2-amine | HCID 43559251 | — |
| Reactant | 5-Cyclopentyl-6-cyclopropylmethoxy-pyridine-2-carboxylic acid | HCID 71087559 | — |
| Product | 5-Cyclopentyl-6-cyclopropylmethoxy-pyridine-2-carboxylic acid [1-methyl-1-(5-methyl-[1,2,4]oxadiazol-3-yl)-ethyl]-amide | HCID 71093575 | — |
Reaction Steps
The title compound was synthesized in analogy to Example 1, using 5-cyclopentyl-6-cyclopropylmethoxy-pyridine-2-carboxylic acid (Example 39 b) and α,α,5-trimethyl-1,2,4-oxadiazole-3-methanamine (CAN 1153831-97-0, Example 33 d) as starting materials, MS (LC/MS): 385.2 [M+H]+.
Provenance & Evidence
| DOI | 10.6084/m9.figshare.5104873.v1 |
|---|---|
| Patent number | US09290451B2 |
| Source dataset | uspto-grants-2016_03 |
| ORD ID | ord-eb7394d0d0964c1fb1f092e98f823590 |
| Source note | uspto-grants-2016_03 |