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HRID928308

反应详情

EQUATION

反应方程式

HRID 928308 的结构方程式

REACTANTS

反应物

2
结构：CC#CC(=O)O
HCID68535

2-Butynoic acid

C4H4O2

结构：Cc1ccnc(NC(=O)c2ccc(-c3nc([C@@H]4CCCN4)n4ccnc(N)c34)cc2)c1
HCID71226355

未命名化合物

2 次

PRODUCTS

生成物

1
结构：CC#CC(=O)N1CCC[C@H]1c1nc(-c2ccc(C(=O)Nc3cc(C)ccn3)cc2)c2c(N)nccn12
HCID71226074

未命名化合物

收率 27.2%

PROCEDURE

实验过程

This compound was prepared, in an analogous manner as described in Example 2, from (S)-4-(8-amino-3-(pyrrolidin-2-yl)imidazo[1,5-a]pyrazin-1-yl)-N-(4-methylpyridin-2-yl)benzamide (intermediate 7) and 2-butynoic acid, to afford the title compound (6.3 mg, 27.2%). Data: UPLC (C) Rt: 1.56 min; m/z 480.3 (M+H)+.

WORKUP

后处理

  1. customThis compound was prepared, in an analogous manner