HCID 63893296, compound → HCID 86715606, compound
Reaction equation
[CH3:1][N:2]([CH3:17])[C:3]1[CH:8]=[CH:7][C:6]([CH:9]([C:11]2[CH:12]=[N:13][CH:14]=[CH:15][CH:16]=2)[OH:10])=[CH:5][CH:4]=1.CN1C(C(C2C=CC=CN=2)O)=CN=C1>>[CH3:1][N:2]([CH3:17])[C:3]1[CH:4]=[CH:5][C:6]([C:9]([C:11]2[CH:12]=[N:13][CH:14]=[CH:15][CH:16]=2)=[O:10])=[CH:7][CH:8]=1Participants
3
Procedure
The title compound was prepared analogously to the method in Intermediate 25: step b using (4-(dimethylamino)phenyl)(pyridin-3-yl)methanol (Intermediate 28: step a) in place of (1-methyl-1H-imidazol-5-yl)(pyridin-2-yl)methanol.
Sources & evidence
- ORD record
- ord-4a9255e53e97472f890279cd682fb225
- Source dataset
- uspto-grants-2016_03
- Patent number
- US09290476B2
Reaction notes
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