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HuagongsheHuagongshe Chemistry Print Report · For research reference only
HRID 985799Generated: October 30, 2026

Azetidine → (+)-2-Azetidin-1-yl-N-(7-[1,4]dioxan-2-yl-4-methoxy-benzothiazol-2-yl)-isonicotinamide

https://huagongshe.com/reaction/985799

Reaction equation

Participants

RoleNameHCIDCharge
ReactantAzetidineHCID 10422—
ReactantCesium carbonateHCID 10796—
Reactant(+)-2-bromo-N-(7-[1,4]dioxan-2-yl-4-methoxy-benzothiazol-2-yl)-isonicotinamideHCID 22507693—
Product(+)-2-Azetidin-1-yl-N-(7-[1,4]dioxan-2-yl-4-methoxy-benzothiazol-2-yl)-isonicotinamideHCID 11487132—

Reaction Steps

From (±)-2-bromo-N-(7-[1,4]dioxan-2-yl-4-methoxy-benzothiazol-2-yl)-isonicotinamide with cesium carbonate and azetidine. ES-MS m/e (%): 427 (M+H+, 100).

Provenance & Evidence

DOI10.6084/m9.figshare.5104873.v1
Patent numberUS06872833B2
Source datasetuspto-grants-2005_03
ORD IDord-37b18456fa254613b68fe20a20c3b0d8
Source noteuspto-grants-2005_03