Glycine → Argininamide

HRID 1761382

Reaktionsgleichung

Reaktionsgleichung von HRID 1761382
[NH2:1][C@@H](C(O)=O)CC1C=CC(O)=CC=1.N[C@@H](C(O)=O)CC1C=CC(OCC)=CC=1.N[C@H](C(O)=O)CC1C=CC=CC=1.N[C@H](C(O)=O)C(C)C.[NH2:49][C@H:50]([C:58]([OH:60])=O)[CH2:51][CH2:52][CH2:53][NH:54][C:55](=[NH:57])[NH2:56].N(C)[C@H](C(O)=O)CCCNC(=N)N.NCC(O)=O>>[NH2:49][C@H:50]([C:58]([NH2:1])=[O:60])[CH2:51][CH2:52][CH2:53][NH:54][C:55](=[NH:57])[NH2:56]

Komponenten

8

Edukt 7

HCID 750Glycine2×HCID 6140L-PhenylalanineHCID 6287L-ValineHCID 71098D-TyrosineHCID 18596379O-Ethyl-D-tyrosineHCID 178418600HCID 178418600, Verbindung2×HCID 178484884HCID 178484884, Verbindung

Produkt 1

HCID 178512843Argininamide

Versuchsvorschrift

A compound of claim 1 in which A is D-Tyr or D-Tyr(Et); B is Phe; C is Val; m, p and q are each 0 or 1; W is a D or L isomer of Pro, Arg or N-MeArg; X is a D or L isomer of Arg or Gly; Y is Gly; and Z is NHR or a D or L isomer of Arg-NH2, provided that X is not Gly when m is 0, and q is 0 if both m and p are 0.

Quellen und Nachweise

ORD-Eintrag
ord-831104fd4ae64dbead2f796a88d85836
Quelldatensatz
uspto-grants-1989_05
Patentnummer
US04826813

Verknüpfte Notizen

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