HuagongsheHuagongshe Chemie-Druckbericht · Nur für Forschungszwecke
1-Benzyl-1H-pyrazole-4-boronic acid → 2-(1-Benzyl-1h-pyrazol-4-yl)-4-{[(2,4-dimethoxy-benzyl)-ethoxycarbonylmethyl-amino]-methyl}-thiazole-5-carboxylic acid ethyl ester
Beteiligte Stoffe
| Rolle | Name | HCID | Einwaage |
|---|---|---|---|
| Edukt | 1-Benzyl-1H-pyrazole-4-boronic acid | HCID 3352881 | — |
| Edukt | 2-Bromo-4-{[(2,4-dimethoxy-benzyl)-ethoxycarbonylmethyl-amino]-methyl}-thiazole-5-carboxylic acid ethyl ester | HCID 68426454 | — |
| Produkt | 2-(1-Benzyl-1h-pyrazol-4-yl)-4-{[(2,4-dimethoxy-benzyl)-ethoxycarbonylmethyl-amino]-methyl}-thiazole-5-carboxylic acid ethyl ester | HCID 68428356 | — |
Reaktionsschritte
Prepared from 2-bromo-4-{[(2,4-dimethoxy-benzyl)-ethoxycarbonylmethyl-amino]-methyl}-thiazole-5-carboxylic acid ethy ester, example 81(b), and 1-benzyl-1H-pyrazole-4-boronic acid under conditions analogous to experimental example 81(c). MS: (+) m/z 579.4 (M+1).
Herkunft & Nachweise
| DOI | 10.6084/m9.figshare.5104873.v1 |
|---|---|
| Patentnummer | US07696223B2 |
| Quelldatensatz | uspto-grants-2010_04 |
| ORD ID | ord-aa1431426e2943b1ae653397f8acf1d7 |
| Quellennotiz | uspto-grants-2010_04 |