4-Nitrobenzoic Acid → 2-bromo-N-(imidazo[1,2-a]pyridin-6-ylmethyl)thiazole-5-carboxamide
Reaktionsgleichung
CC(C)[CH2:3][CH2:4][NH2:5].[Br:7][C:8]1[S:9][C:10]([C:13]([NH2:15])=[O:14])=[CH:11][N:12]=1.[N+:16]([C:19]1[CH:27]=[CH:26][C:22]([C:23](O)=O)=[CH:21]C=1)([O-])=O>>[Br:7][C:8]1[S:9][C:10]([C:13]([NH:15][CH2:23][C:22]2[CH:26]=[CH:27][C:19]3[N:16]([CH:3]=[CH:4][N:5]=3)[CH:21]=2)=[O:14])=[CH:11][N:12]=1Komponenten
4
Versuchsvorschrift
The title compound was prepared as described in Example 1A, substituting imidazo[1,2-a]pyridin-6-ylmethanamine for 3-methylbutan-1-amine and 2-bromothiazole-5-carboxamide for 4-nitrobenzoic acid.
Quellen und Nachweise
- ORD-Eintrag
- ord-6a6171473f4a4eafa53f13cc26974e3c
- Quelldatensatz
- uspto-grants-2015_11
- Patentnummer
- US09187472B2
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