(4-Methoxyphenyl)boronic acid → HCID 18448288, compound

Reaction equation

[CH3:1][O:2][C:3]1[CH:8]=[CH:7][C:6](B(O)O)=[CH:5][CH:4]=1.Br[C:13]1[C:14]([CH3:39])=[C:15]([N:19]([CH2:24][C:25]2[CH:37]=[CH:36][C:28]([O:29][CH2:30][C:31]([O:33]CC)=[O:32])=[C:27]([CH3:38])[CH:26]=2)[CH2:20][CH2:21][O:22][CH3:23])[CH:16]=[CH:17][CH:18]=1>>[CH3:23][O:22][CH2:21][CH2:20][N:19]([CH2:24][C:25]1[CH:37]=[CH:36][C:28]([O:29][CH2:30][C:31]([OH:33])=[O:32])=[C:27]([CH3:38])[CH:26]=1)[C:15]1[C:14]([CH3:39])=[C:13]([C:6]2[CH:7]=[CH:8][C:3]([O:2][CH3:1])=[CH:4][CH:5]=2)[CH:18]=[CH:17][CH:16]=1

Participants

Reactant 2

HCID 201262(4-Methoxyphenyl)boronic acid

HCID 58622864HCID 58622864, compound

Product 1

HCID 18448288HCID 18448288, compound

Procedure

Prepared from 4-methoxyphenylboronic acid and ethyl (4-{[(3-bromo-2-methylphenyl)(2-methoxyethyl)amino]methyl}-2-methylphenoxy)acetate using the procedure described for Example 25 (Method A).

Sources & evidence

ORD record: ord-0db6db38b1584e4ebdbd144615e155db
Source dataset: uspto-grants-2007_04
DOI: 10.6084/m9.figshare.5104873.v1
Patent number: US07199239B2

Reaction notes

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