Cl.Cl.[NH2:3][NH2:4].C(O/[CH:8]=[CH:9]/[C:10](=O)[C:11]([F:14])([F:13])[F:12])C.C(OCC)(=O)C.CCCCCC>C(O)C>[F:12][C:11]([F:14])([F:13])[C:10]1[CH:9]=[CH:8][NH:4][N:3]=1Hydrazine dihydrochloride (225 g, 2.14 mol) in ethanol (1400 mL) was stirred well. TEA (185.4 mL, 1.34 mol) was added drop wise for 45 min at ambient temperature. Then (E)-4-ethoxy-1,1,1-trifluorobut-3-en-2-one (225 g, crude) was added drop wise at room temperature and the overall reaction mixture was refluxed overnight. Progress of the reaction was monitored by TLC (20% ethyl acetate/hexane, Rf˜0.4). On completion of the reaction, ethanol was distilled off completely, residue was taken in ice water (500 mL) and the product extracted with ethyl acetate (2×400 mL). Combined extract was washed with ice water (300 mL), dried over sodium sulfate and concentrated under reduced pressure to yield 3-(trifluoromethyl)-1H-pyrazole as a off white solid (175 g, crude).
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