Morpholine → HCID 67153308, compound
Reaction equation
CS(OC[CH2:7][O:8][C:9]1[CH:14]=[CH:13][CH:12]=[C:11]([C:15]2[N:19]([C:20]3[CH:25]=[CH:24][CH:23]=[C:22]([Cl:26])[CH:21]=3)[N:18]=[C:17]([C:27]([N:29]3[CH2:33][C:32](=[O:34])[NH:31][CH2:30]3)=[O:28])[CH:16]=2)[CH:10]=1)(=O)=O.N1CCOCC1.[CH:41]([OH:43])=[O:42].ClC1C=C(N2C(C3C=CC=C(OCCCN(C)C)C=3)=C[C:53]([C:69]([N:71]3[CH2:75][C:74](=[O:76])N[CH2:72]3)=O)=N2)C=CC=1>O1CCCC1>[CH:41]([OH:43])=[O:42].[Cl:26][C:22]1[CH:21]=[C:20]([N:19]2[C:15]([C:11]3[CH:12]=[CH:13][CH:14]=[C:9]([O:8][CH2:7][CH2:72][N:71]4[CH2:69][CH2:53][O:76][CH2:74][CH2:75]4)[CH:10]=3)=[CH:16][C:17]([C:27]([N:29]3[CH2:33][C:32](=[O:34])[NH:31][CH2:30]3)=[O:28])=[N:18]2)[CH:25]=[CH:24][CH:23]=1Participants
5
Reactant 3
Product 1
Reagents, catalysts & solvents 1
Procedure
The preparation of the title compound takes place starting from the compound of Example 121A and morpholine without the addition of tetrahydrofuran in analogy to the synthesis of the compound of Example 29. 47 mg (43% of theory) of the title compound are obtained.